AnnoTitoloTipo MIUR
2026Semi-Synthetic H2S Releasing Compounds with Antioxidant and Vasorelaxant Properties
(ACS MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2025Heme oxygenase 1 inhibitor discovery and formulation into nanostructured lipid carriers as potent and selective treatment against triple negative metastatic breast cancer
(INTERNATIONAL JOURNAL OF PHARMACEUTICS)
Articolo in rivista
2024Combination of heme oxygenase-1 inhibitors and temozolomide to improve the anticancer effect in glioblastoma
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY REPORTS)
Articolo in rivista
2024Evaluation of the anticancer effects exerted by 5-fluorouracil and heme oxygenase-1 inhibitor hybrids in HTC116 colorectal cancer cells
(JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY)
Articolo in rivista
2024Synthesis and in Vitro Evaluation of CAPE Derivatives as Ferroptosis Inducers in Triple Negative Breast Cancer
(ACS MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2023Discovery of SI 1/20 and SI 1/22 as Mutual Prodrugs of 5-Fluorouracil and Imidazole-Based Heme Oxygenase 1 Inhibitor with Improved Cytotoxicity in DU145 Prostate Cancer Cells
(CHEMMEDCHEM)
Articolo in rivista
2023In vitro and in silico analysis of imatinib analogues as anti- Trypanosoma cruzi drug candidates
(PARASITOLOGY)
Articolo in rivista
2023Novel Heme Oxygenase-1 Inducers Palliate Inflammatory Pain and Emotional Disorders by Regulating NLRP3 Inflammasome and Activating the Antioxidant Pathway
(ANTIOXIDANTS)
Articolo in rivista
2023The Inhibition of Neuropathic Pain Incited by Nerve Injury and Accompanying Mood Disorders by New Heme Oxygenase-1 Inducers: Mechanisms Implicated
(ANTIOXIDANTS)
Articolo in rivista
2022CAPE and its synthetic derivative VP961 restore BACH1/NRF2 axis in Down Syndrome
(FREE RADICAL BIOLOGY & MEDICINE)
Articolo in rivista
2022Heme Oxygenase Modulation Drives Ferroptosis in TNBC Cells
(INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES)
Articolo in rivista
2022Novel Tyrosine Kinase Inhibitors to Target Chronic Myeloid Leukemia
(MOLECULES)
Articolo in rivista
2022Structure-activity relationships of mixed σ1R/σ2R ligands with antiproliferative and anticancer effects
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2021A computer-aided approach to identify novel Leishmania major protein disulfide isomerase inhibitors for treatment of leishmaniasis
(JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN)
Articolo in rivista
2021Combination of heme oxygenase-1 inhibition and sigma receptor modulation for anticancer activity
(MOLECULES)
Articolo in rivista
2021Development of New Benzylpiperazine Derivatives as σ1Receptor Ligands with in Vivo Antinociceptive and Anti-Allodynic Effects
(ACS CHEMICAL NEUROSCIENCE)
Articolo in rivista
2021Discovery of Novel Acetamide-Based Heme Oxygenase-1 Inhibitors with Potent in Vitro Antiproliferative Activity
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2021Glucose-impaired Corneal Re-epithelialization Is Promoted by a Novel Derivate of Dimethyl Fumarate
(ANTIOXIDANTS)
Articolo in rivista
2021Growing the molecular architecture of imidazole-like ligands in HO-1 complexes
(BIOORGANIC CHEMISTRY)
Articolo in rivista
2021Mutual Prodrugs of 5-Fluorouracil: From a Classic Chemotherapeutic Agent to Novel Potential Anticancer Drugs
(CHEMMEDCHEM)
Articolo in rivista
2021Novel mutual prodrug of 5-fluorouracil and heme oxygenase-1 inhibitor (5-FU/HO-1 hybrid): design and preliminary in vitro evaluation
(JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY)
Articolo in rivista
2021Potential health benefits of a pomegranate extract, rich in phenolic com-pounds, in intestinal inflammation
(CURRENT NUTRITION & FOOD SCIENCE)
Articolo in rivista
2021Recent Advances in the Development of Sigma Receptor Ligands as Cytotoxic Agents: A Medicinal Chemistry Perspective
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2020Chromatograpic resolution of phenylethanolic-azole racemic compounds highlighted stereoselective inhibition of heme oxygenase-1 by (R)-enantiomers
(BIOORGANIC CHEMISTRY)
Articolo in rivista
2020Identification of a potent heme oxygenase-2 (HO-2) inhibitor by targeting the secondary hydrophobic pocket of the HO-2 western region
(BIOORGANIC CHEMISTRY)
Articolo in rivista
2020New arylethanolimidazole derivatives as HO-1 inhibitors with cytotoxicity against MCF-7 breast cancer cells
(INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES)
Articolo in rivista
2020Non-competitive heme oxygenase-1 activity inhibitor reduces non-small cell lung cancer glutathione content and regulates cell proliferation
(MOLECULAR BIOLOGY REPORTS)
Articolo in rivista
2020Novel heme oxygenase-1 (Ho-1) inducers based on dimethyl fumarate structure
(INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES)
Articolo in rivista
2020Novel N-Substituted Benzomorphan-Based Compounds: From MOR-Agonist/DOR-Antagonist to Biased/Unbiased MOR Agonists
(ACS MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2020Synthesis and Molecular Modelling Studies of New 1,3-Diaryl-5-Oxo-Proline Derivatives as Endothelin Receptor Ligands
(MOLECULES)
Articolo in rivista
2019Fourfold filtered statistical/computational approach for the identification of imidazole compounds as HO-1 inhibitors from natural products
(MARINE DRUGS)
Articolo in rivista
2019Ginseng and heme oxygenase-1: The link between an old herb and a new protective system
(FITOTERAPIA)
Articolo in rivista
2019Heme Oxygenase Inhibition Sensitizes Neuroblastoma Cells to Carfilzomib
(MOLECULAR NEUROBIOLOGY)
Articolo in rivista
2019Heme Oxygenase-1 Inhibition Sensitizes Human Prostate Cancer Cells towards Glucose Deprivation and Metformin-Mediated Cell Death
(INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES)
Articolo in rivista
2019Heme Oxygenase-2 (HO-2) as a therapeutic target: Activators and inhibitors
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2019HO-1 INHIBITION POTENTIATES METFORMIN ANTINEOPLASTIC EFFECTS IN HUMAN PROSTATE CANCER CELLS UNDER LOW GLUCOSE CONCENTRATIONPoster
2019Nanotechnological Approach to Increase the Antioxidant and Cytotoxic Efficacy of Crocin and Crocetin
(PLANTA MEDICA)
Articolo in rivista
2019Progress in the development of more effective and safer analgesics for pain management
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2019Progress in the development of selective heme oxygenase-1 inhibitors and their potential therapeutic application
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2019Protective Effects of Caffeic Acid Phenethyl Ester (CAPE) and Novel Cape Analogue as Inducers of Heme Oxygenase-1 in Streptozotocin-Induced Type 1 Diabetic Rats
(INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES)
Articolo in rivista
2019Synthesis, in vitro and in silico studies of HO-1 inducers and lung antifibrotic agents
(FUTURE MEDICINAL CHEMISTRY)
Articolo in rivista
2019Synthesis, in vitro and in vivo characterization of new benzoxazole and benzothiazole-based sigma receptor ligands
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2019[1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2018Caratterizzazione chimico-fisica ed attività antiossidante in vitro del triestere trans-resveratrolotrolox.Abstract in Atti di convegno
2018Development of new HO-1 inhibitors by a thorough scaffold-hopping analysis
(BIOORGANIC CHEMISTRY)
Articolo in rivista
2018Effects of Polyphenolic Derivatives on Heme Oxygenase-System in Metabolic Dysfunctions
(CURRENT MEDICINAL CHEMISTRY)
Articolo in rivista
2018Identification of Potentially Potent Heme Oxygenase 1 Inhibitors through 3D-QSAR Coupled to Scaffold-Hopping Analysis
(CHEMMEDCHEM)
Articolo in rivista
2018New homo and hetero bis-arylpiperazine and bis-benzylpiperazine derivatives as 5-HT7R selective ligands: design and synthesisAbstract in Atti di convegno
2018Novel structural insight into inhibitors of heme oxygenase-1 (ho-1) by new imidazole-based compounds: Biochemical and in vitro anticancer activity evaluation
(MOLECULES)
Articolo in rivista
2018Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitors
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2018Potholing of the hydrophobic heme oxygenase-1 western region for the search of potent and selective imidazole-based inhibitorsAbstract in Atti di convegno
2018Structure-Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2018Synthesis and in vitro antioxidant activity of a novel idebenone ester with pyroglutamic acid.Abstract in Atti di convegno
2018Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2018Therapeutic Potential of Caffeic Acid Phenethyl Ester (CAPE) in Diabetes.
(CURRENT MEDICINAL CHEMISTRY)
Articolo in rivista
2017ATTIVITÀ ANTIOSSIDANTE IN VITRO DI DERIVATI DELL’IDEBENONEAbstract in Atti di convegno
2017Comprehensive data on a 2D-QSAR model for Heme Oxygenase isoform 1 inhibitors
(DATA IN BRIEF)
Articolo in rivista
2017Effects of Novel Nitric Oxide-Releasing Molecules against Oxidative Stress on Retinal Pigmented Epithelial Cells
(OXIDATIVE MEDICINE AND CELLULAR LONGEVITY)
Articolo in rivista
2017Heme Oxygenase Database (HemeOxDB) and QSAR Analysis of Isoform 1 Inhibitors
(CHEMMEDCHEM)
Articolo in rivista
2017Heme Oxygenase-1: A new druggable target in the management of chronic and acute myeloid leukemia
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2017In vitro antioxidant activity of idebenone derivative-loaded solid lipid nanoparticles
(MOLECULES)
Articolo in rivista
2017New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2017Novel Caffeic Acid Phenethyl Ester (Cape) Analogues as Inducers of Heme Oxygenase-​1
(CURRENT PHARMACEUTICAL DESIGN)
Articolo in rivista
2017Recent advances in drug discovery of phototherapeutic non-porphyrinic anticancer agents
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2017Role of the Nrf2/HO-1 axis in bronchopulmonary dysplasia and hyperoxic lung injuries
(CLINICAL SCIENCE)
Articolo in rivista
2017Synthesis and experimental validation of new designed heterocyclic compounds with antiproliferative activity versus breast cancer cell lines MCF-7 and MDA-MB-231
(JOURNAL OF CHEMISTRY)
Articolo in rivista
2017Synthesis of Novel Benzylpiperazine Derivatives as Ligands for the σ1 ReceptorAbstract in Atti di convegno
2017Targeting Heme Oxygenase-1 to Overcome Imatinib Resistance in Chronic Myeloid LeukemiaAbstract in Atti di convegno
2016Antiangiogenic Effect of (±)-Haloperidol Metabolite II Valproate Ester [(±)-MRJF22] in Human Microvascular Retinal Endothelial Cells
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2016Design and synthesis of new homo and hetero bis-piperazinyl-1- propanone derivatives as 5-HT7R selective ligands over 5-HT1AR
(BIOORGANIC & MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2016Haloperidol Metabolite II Valproate Ester: Antiangiogenic Activity in Human Microvascular Retinal Endothelial CellsAbstract in Atti di convegno
2016HALOPERIDOL METABOLITE II VALPROATE ESTER: ANTIANGIOGENIC ACTIVITY IN HUMAN MICROVASCULAR RETINAL ENDOTHELIAL CELLSPoster
2016Heme Oxygenase-1 Inhibition: A Novel Strategy for the Design of Azole-Based Antitumour AgentsAbstract in Atti di convegno
2016Novel Caffeic Acid Phenethyl Ester (CAPE) Analogues as Inducers of Heme Oxygenase-1Abstract in Atti di convegno
2016Novel selective ligands for the serotonergic 5-HT7 receptor: tricyclic derivatives Bearing the pyrimido-4(3H)-one ringAbstract in Atti di convegno
2016Rescuing Abandoned Molecules as Nav1.7 and PCSK9 Inhibitors
(JOURNAL OF ADVANCES IN MEDICAL AND PHARMACEUTICAL SCIENCES)
Articolo in rivista
2015An alpha1-adrenergic receptor ligand repurposed as a potent antiproliferative agent for head and neck squamous cell carcinoma
(RSC ADVANCES)
Articolo in rivista
2015Analysis of mechanisms for memory enhancement using novel and potent 5-HT1A receptor ligands
(EUROPEAN NEUROPSYCHOPHARMACOLOGY)
Articolo in rivista
2015CAFFEIC ACID PHENETHYL ESTER (CAPE) DERIVATIVES AS NOVEL HEME OXYGENASE-1 INDUCERSContributo in Atti di convegno
2015Caffeic Acid Phenethyl Ester (CAPE) derivatives as novel heme oxygenase-1 inducers.Poster
2015Caffeic acid phenetyl ester (CAPE) derivatives as novel heme oxygenase-1 inducersContributo in Atti di convegno
2015Effects of novel hybrids of caffeic acid phenethyl ester and NSAIDs on experimental ocular inflammation
(EUROPEAN JOURNAL OF PHARMACOLOGY)
Articolo in rivista
2015How does binding of imidazole-based inhibitors to heme oxygenase-1 influence their conformation? Insights combining crystal structures and molecular modelling
(ACTA CRYSTALLOGRAPHICA. SECTION B, STRUCTURAL SCIENCE, CRYSTAL ENGINEERING AND MATERIALS)
Articolo in rivista
2015New 5-Ht7 Receptor Ligands As Potential Antidepressant Agents.Poster
2015Novel imidazole derivatives as heme oxygenase-1 (HO-1) and heme oxygenase-2 (HO-2) inhibitors and their cytotoxic activity in human-derived cancer cell lines
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2015Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT1A and 5-HT7 receptor ligands
(BIOORGANIC & MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2015Synthesis and Endothelin Receptors Binding Affinity of New 1,3,5- Substituted Pyrrole-2-Carboxylic Acid Derivatives
(MEDICINAL CHEMISTRY)
Articolo in rivista
2014Antioxidant Activity and Phenolic Content of Microwave-Assisted Solanum melongena Extracts
(THE SCIENTIFIC WORLD JOURNAL)
Articolo in rivista
2014High affinity ligands and potent antagonists for the alpha1D-adrenergic receptor. Novel 3,8-disubstituted [1]benzothieno[3,2-d]pyrimidine derivatives
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2014New alkylpiperazines as 5-HT7R ligandsContributo in Atti di convegno
2014New alkylpiperazines as 5-HT7R ligandsAbstract in Atti di convegno
2014New alkylpiperazines as 5-HT7R ligandsPoster
2014Structure-activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2014Thieno[3,2-d]pyrimidine as a scaffold for 5-HT7 receptor ligandsPoster
2014Thieno[3,2-d]pyrimidine as a scaffold for 5-HT7 receptor ligandsAbstract in Atti di convegno
2013A focus on Heme Oxygenase-1 (HO-1) inhibitors
(CURRENT MEDICINAL CHEMISTRY)
Articolo in rivista
2013Antitumor properties of substituted (alpha E)-alpha-(1H-indol-3-ylmethylene)benzeneacetic acids or amides
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2013Evaluation of novel aryloxyalkyl derivatives of imidazole and 1,2,4-triazole as heme oxygenase-1 (HO-1) inhibitors and their antitumor properties
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2013Evaluation of novel aryloxyalkyl derivatives of imidazole and 1,2,4-triazole as Heme Oxygenase-1 inhibitors and their antitumor propertiesAbstract in Atti di convegno
2013New thienopyrimidine and quinazoline derivatives as potential 5-HT7 receptor ligandsContributo in Atti di convegno
2013New thienopyrimidine and quinazoline derivatives as potential 5-HT7 receptor ligands.Abstract in Atti di convegno
2013Thieno[3,2-d]pyrimidin-4(3H)-one derivatives as novel ligands for the 5-HT7 receptorAbstract in Atti di convegno
2013Thieno[3,2-d]pyrimidin-4(3H)-one derivatives as novel 5-HT7 receptorContributo in Atti di convegno
2013Thieno[3,2-d]pyrimidin-4(3H)-one derivatives as novel 5-HT7 receptor ligandsContributo in Atti di convegno
2012Binding Mode Analysis and Pharmacophore Development for Imidazole Derivatives as Heme Oxygenase (HO) InhibitorsContributo in Atti di convegno
2012(E)-alfa-[[(5-Substituted)1H-indol- 3-yl]methylene]benzeneacetic acid and amide derivatives: synthesis, characterization, and evaluation of in vitro antiproliferative activityPoster
2012(E)-alfa-[[(5-substituted)1H-indol-3-yl]methylene]benzeneacetic acid and amide derivatives: synthesis, characterization, and evaluation of in vitro antiproliferative activityAbstract in Atti di convegno
2012(E)-alpha-[[(5-Substituted)1H-indol-3-yl]methylene]benzeneacetic Acid and Amide Derivatives: Synthesis, Characterization, and Evaluation of in vitro Antiproliferative ActivityContributo in Atti di convegno
2012Evaluation of Imidazole-Based Compounds as Heme Oxygenase-1 Inhibitors
(CHEMICAL BIOLOGY & DRUG DESIGN)
Articolo in rivista
2012Evaluation of Novel Imidazole- and 1,2,4 Triazole-based Compounds as Heme Oxygenase-1 (HO-1) InhibitorsContributo in Atti di convegno
2012Evaluation of Novel Imidazole- and 1,2,4 Triazole-based Compounds as Heme Oxygenase-1 (HO-1) Inhibitors.Poster
2012(E)-?-[[(5-Substituted)1H-indol-3-yl]methylene]benzeneacetic Acid and Amide Derivatives: Synthesis, Characterization, and Evaluation of in vitro Antiproliferative ActivityContributo in Atti di convegno
2012Imidazole Derivatives as Heme Oxygenase-1 InhibitorsPoster
2012Imidazole Derivatives as Heme Oxygenase-1 InhibitorsAbstract in Atti di convegno
2012Imidazole Derivatives as Heme Oxygenase-1 InhibitorsContributo in Atti di convegno
2012Novel inhibitors of nitric oxide synthase with antioxidant properties
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2011A New benzoxazolone and benzothiazolone derivatives as potential 5-HT7 receptor ligandsAbstract in Atti di convegno
2011New benzoxazolone and benzothiazolone derivatives as potential 5-HT7 receptor ligands.Contributo in Atti di convegno
2011NEW BENZOXAZOLONE AND BENZOTHIAZOLONE DERIVATIVES AS POTENTIAL 5-HT7 RECEPTOR LIGANDSAbstract in Atti di convegno
2011Novel 4-phenylpiperidine-2,6-dione derivatives. Ligands for alpha1-adrenoceptor subtypes.
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2011Synthesis and molecular modeling of 1H-pyrrolopyrimidine-2,4-dione derivatives as ligands for the alpha1-adrenoceptors
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2010Novel [1]benzothieno[[3,2-d]pyrimidin-4(3H)-ones. Ligands for the 5-HT7 receptor
(DRUGS OF THE FUTURE)
Contributo in Atti di convegno
2010Serotonin 5-HT3 and 5-HT4 Ligands: An Update of Medicinal Chemistry Research in the Last Few Years
(CURRENT MEDICINAL CHEMISTRY)
Articolo in rivista
2009New benzooxazole and benzothiazole derivatives as potential 5-HT7 receptor ligandsContributo in Atti di convegno
2009New benzoxazole and benzothiazole derivatives as potential 5-HT7 receptor ligandsContributo in Atti di convegno
2008In search of the Magic Bullets: Discover of RN5 and its Structural Modifications for Targeting Selectively alpha 1 AdrenoceptorsContributo in Atti di convegno
2008In search of the Magic Bullets: Discover of RN5 and its Structural Modifications for Targeting Selectively alpha 1 AdrenoceptorsAbstract in Atti di convegno
2008Molecular modeling explains differences in binding affinity of new potent and selective 5-HT1A ligands: arylpiperazinylalkylthiobenzoxazole derivatives. The Sixth Multidisciplinary Conference on Drug ResearchAbstract in Atti di convegno
2008New compounds controlling NO overproductionContributo in volume (Capitolo o Saggio)
2008New thienopyrimidine derivatives as potential 5-HT7 receptor ligandsAbstract in Atti di convegno
2008New thienopyrimidine derivatives as potential 5-HT7 receptor ligandsContributo in Atti di convegno
2008Simultaneus Determination of Catechins, Rutin, and Gallic Acid in Cistus Species Extracts by HPLC with Diode Array Detection
(JOURNAL OF CHROMATOGRAPHIC SCIENCE)
Articolo in rivista
2008Synthesis and endothelin receptor binding affinity of a novel class of 2-substituted-4-aryl-3-quinolinecarboxylic acid derivatives
(MEDICINAL CHEMISTRY)
Articolo in rivista
2008Synthesis and receptor binding of new thieno[2,3-d]pyrimidines as selective ligands of 5-HT3 receptors
(ARCHIV DER PHARMAZIE)
Articolo in rivista
2008Synthesis of new arylpiperazinylalkylthiobenzimidazole, benzothiazole, or benzoxazole, derivatives as potent and selective 5-HT1A serotonin receptor ligands
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
2007Arylpiperazinylalkylthio benzothiazole or benzoxazole as selective 5-HT1A serotonin receptor ligandsContributo in Atti di convegno
2007Arylpiperazinylalkylthio benzothiazole or benzoxazole derivatives as selective 5-HT1A serotonin receptor ligandsContributo in Atti di convegno
2007Arylpiperazinylalkylthio benzothiazole or benzoxazole derivatives as selective 5-HT1A serotonin receptor ligandsAbstract in Atti di convegno
2007Benzothieno[3,2-d]pyrimidine ligands with high affinity for human alpha1-adrenergic receptor subtypesAbstract in Atti di convegno
2007Inhibition of Human Leucocyte Elastase by Novel Thieno-1,3-oxazin-4-ones and Thieno-1,3-thioxazin-4-ones
(LETTERS IN DRUG DESIGN & DISCOVERY)
Articolo in rivista
2007Nuovi Arilpiperazinilalchilpirrolopirimidindioni come ligandi potenti e selettivi per i recettori α1-adrenergiciAbstract in Atti di convegno
2007Synthesis and Binding Properties of New Endothelin Receptor Ligands
(LETTERS IN DRUG DESIGN & DISCOVERY)
Articolo in rivista
2007SYNTHESIS OF 1,2,4-TRIAZOLE DERIVATIVES: BINDING PROPERTIES ON ENDOTHELIN RECEPTORS
(MEDICINAL CHEMISTRY)
Articolo in rivista
20075-HT7 receptor ligands: recent developments and potential therapeutic applications
(MINI-REVIEWS IN MEDICINAL CHEMISTRY)
Articolo in rivista
2006Imidazole derivatives as antioxidants and selective inhibitors of nNOS
(NITRIC OXIDE)
Articolo in rivista
2006New Pyrimido[5,4-b]indoles and [1]Benzothieno[3,2-d]pyrimidines. High Affinity Ligands for the a 1 - Adrenoceptor Subtypes
(BIOORGANIC & MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2006New 1,2,3,9-tetrahydro-4H-carbazol-4-one derivatives: Analogues of HEAT as ligands for the alpha(1)-adrenergic receptor subtypes
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2006Novel arylpiperazine ligands with high affinity for alpha1-adrenergic receptor subtypesAbstract in Atti di convegno
2006Synthesis and binding properties of new endothelin receptor ligandsAbstract in Atti di convegno
2006Synthesis and endothelin receptor binding affinity of a novel class of 2-Substituted-4-aryl-3-quinolinecarboxylic Acid DerivativesAbstract in Atti di convegno
20063-Arylpiperazinylethyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione derivatives as novel, high affinity and selective alpha1-adrenoceptor ligands
(BIOORGANIC & MEDICINAL CHEMISTRY LETTERS)
Articolo in rivista
2005A Facile Synthesis of New 2-carboxamido-3-carboxythiophene and 4,5,6,7-tetrahydro-2-carboxyamido-3-carboxythieno[2,3-c]pyridine Derivatives as Potential Endothelin Receptors Ligands
(IL FARMACO)
Articolo in rivista
2005Design and Synthesis of New 3-Aryl-5-oxoprolines as Potential Ligands for Human Cloned Endothelin ReceptorsContributo in Atti di convegno
2005Design and Synthesis of Novel Potential Ligands for Endothelin ReceptorsContributo in Atti di convegno
2005Design and synthesis of novel potential ligands for endothelin receptorsContributo in Atti di convegno
2005Novel (E)-alpha-[(1H-indol-3-yl)methylene]benzeneacetic Acids as Endothelin Receptor Ligands.
(IL FARMACO)
Articolo in rivista
2005SIMULTANEOUS DETERMINATION OF CATECHINS, RUTIN, AND GALLIC ACID IN CISTUS SPECIES EXTRACTS BY HPLC WITH DIODE ARRAY DETECTIONContributo in Atti di convegno
2005Synthesis and endothelin receptor binding affinity of a novel class of (E)-alpha-[[(5-phenylmethoxy)-1H-indol-3-yl]methylene]benzeneacetic acidsAbstract in Atti di convegno
2005Synthesis of 1,3,5-substituted-pyrroles as potential endhotelin receptor ligandsAbstract in Atti di convegno
2005Synthesis of 3-arylpiperazinylalkylpyrrolo[3,2-d]pyrimidine-2,4-dione derivatives as novel, potent, and selective alpha(1)-adrenoceptor ligands.
(JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
20053-Arylpiperazynilalkyl-1H-pyrrolo[2,3-d]pyrimidine-2,4(3H,7H)-dione derivatives: as novel, potent and selective alpha1-adrenoceptor ligandsAbstract in Atti di convegno
2004Acidi (E)-alfa-[(1-H-indol-3-il)metilene]benzeneacetici. Una nuova classe di ligandi per i recettori delle endotelineContributo in Atti di convegno
2004Acidi (E)-alfa-[(1H-indol-3-il)metilene]benzeneacetici: una nuova classe di ligandi per i recettori delle endotelineAbstract in Atti di convegno
2004ACIDI (E)-a-[(1H-INDOL-3-IL)METILENE]BENZENEACETICI: UNA NUOVA CLASSE DI LIGANDI PER I RECETTORI DELLE ENDOTELINEContributo in Atti di convegno
2004Acidi (E)-[(1H-Indol-3-il)metilene]benzeneacetici: una Nuova Classe di Ligandi per i Recettori delle EndotelineContributo in Atti di convegno
2004Ligandi per le sottoclassi del recettore alfa1-adrenergico. Nuovi derivati benzotieno[3,2-d]pirimidin-(1H,3H)2,4-dionici-8-sostituitiAbstract in Atti di convegno
2004Novel antagonists for α1-adrenoceptor subtypes
(EXPERT OPINION ON THERAPEUTIC PATENTS)
Articolo in rivista
2004Sintesi di 1,2,4 Triazoli come Ligandi per i Recettori delle EndotelineContributo in Atti di convegno
2004Sintesi di 1,2,4 triazoli come ligandi per i recettori delle endotelineAbstract in Atti di convegno
2004Synthesis of new 5-phenyl[1,2,4]triazole derivatives as ligands for the 5-HT1A serotonin receptor
(ARKIVOC)
Articolo in rivista
20043-ARILPIPERAZINILALCHILPIRROLO[3,2-d]PIRIMIDIN-2,4-DIONE: UNA NUOVA CLASSE DI LIGANDI POTENTI ED ALTAMENTE SELETTIVI PER I RECETTORI a 1-ADRENERGICIContributo in Atti di convegno
20043-Arilpiperazinilalchilpirrolo[3,2-d]pirimidin-2,4-dione: una Nuova Classe di Ligandi Potenti ed Altamente Selettivi per i Recettori alfa1 AdrenergiciContributo in Atti di convegno
20043-Arilpiperazinilalchilpirrolo[3,2-d]pirimidin-2,4-dioni: una nuova classe di ligandi potenti e selettivi per il recettori alfa1-adrenergiciContributo in Atti di convegno
2003Benzimidazole, benzoxazole and benzothiazole derivatives as 5-HT1A serotonin receptor ligandsContributo in Atti di convegno
2003DOSAGGIO DI CATECHINE IN ESTRATTI ACQUOSI DI CISTUS INCANUS L. E CISTUS MONSPELIENSIS LContributo in Atti di convegno
2003Novel inhibitors of neuronal nitric oxide synthase
(EXPERIMENTAL BIOLOGY AND MEDICINE)
Articolo in rivista
2003Searching for novel endothelin receptor ligandsContributo in Atti di convegno
2003Searching for Novel Endothelin Receptors LigandsContributo in Atti di convegno
2002Novel imidazole derivatives as selective nNOS inhibitorsContributo in Atti di convegno
2002NUOVI INIBITORI DELLA OSSIDO NITRICO SINTETASIContributo in Atti di convegno
2002Progress in the development of selective nitric oxide synthase (NOS) inhibitors
(CURRENT PHARMACEUTICAL DESIGN)
Articolo in rivista
2002SINTESI DI LIGANDI SELETTIVI PER I RECETTORI alfa1- ADRENERGICIContributo in Atti di convegno
2002SINTESI DI LIGANDI SELETTIVI PER I RECETTORI alfa1-ADRENERGICIContributo in Atti di convegno
2002SINTESI DI LIGANDI SELETTIVI PER I RECETTORI a1-ADRENERGICIContributo in Atti di convegno
2002V. Sorrenti, C. Di Giacomo, L. Salerno, M.A. Siracusa, F. Guerrera, and A. Vanella Novel imidazole derivatives as selective nNOS inhibitorsContributo in Atti di convegno
2002[1,2,4]Triazole derivatives as 5-HT1A serotonin receptor ligands
(BIOORGANIC & MEDICINAL CHEMISTRY)
Articolo in rivista
2001Inhibition of Neuronal Nitric Oxide Synthase by N-Phenacyl Imidazoles
(NITRIC OXIDE)
Articolo in rivista
2001INHIBITION OF NEURONAL NITRIC-OXIDE SYNTHASE (NOS) BY N-PHENACYLAZOLESContributo in Atti di convegno
2001IS-67: A NEW ISOTHIAZOLE WITH A BROAD ANTIVIRAL SPECTRUMContributo in Atti di convegno
2000DI-SUBSTITUTED IMIDAZOLES AS INHIBITORS OF NEURONAL NITRIC OXIDE SYNTHASEContributo in Atti di convegno
2000N-Phenacyl imidazoles as nNos inhibitorsContributo in Atti di convegno
1999Isothiazole derivatives as novel HIV replication inhibitors.Contributo in Atti di convegno
1999N-subsituted imidazoles as inhibitors of nitric oxide synthase: a preliminary screening
(PHARMAZIE)
Articolo in rivista
1999N-substuted-imidazoles as inhibitors of nitric oxide synthase: a preliminary screening.
(PHARMAZIE)
Articolo in rivista
1999Synthesis and Biological Activity of 1-, 2- or 3-Substituted Benzothieno[2,3-d]triazole Derivatives Structurally related to Trazodone.
(JOURNAL OF HETEROCYCLIC CHEMISTRY)
Articolo in rivista
1999Synthesis of novel 4,5-diphenylthiazole derivatives as potential acylCoA:cholesterol O-acyltransferase inhibitors
(PHARMAZIE)
Articolo in rivista
19991-[(aryloxy)alkyl]-1H-imidazoles as inhibitors of neuronal nitric oxide synthase.
(PHARMACY AND PHARMACOLOGY COMMUNICATIONS)
Articolo in rivista
19991-[(Aryloxy)alkyl]-1H-imidazoles as selective inhibitors of neuronal nitric oxide synthase.Contributo in Atti di convegno
19994-Isothiazole carbonitriles active against measles virusContributo in Atti di convegno
1998Isothiazole derivatives as potent antiadenovirus agentsContributo in Atti di convegno
1998Selective inhibition of neuronal nitric oxide synthase by imidazole derivatives.Contributo in Atti di convegno
1998Synthesis and antiviral activity of new 3-(dialkylamino)-5-phenyl-4-isothiazole-carbonitrilesContributo in Atti di convegno
19983-Methylthio-5-(4-ots)-phenyl-4-isothiazolecarbonitrile (IS-44): a new potential HRV capsid-binderContributo in Atti di convegno
1997Inhibition of nitric oxide synthase (NOS) by some N-substituted imidazoles.Contributo in Atti di convegno
1997Isoxazoles with antiviral activityContributo in Atti di convegno
1997Synthesis and pharmacological evaluation of benzothieno and [1]pyridothieno [2,3-d]triazole derivatives as antagonists at NK-1 receptorsContributo in Atti di convegno
1996Isothiazoles as potent and broad spectrum antiviral agentsContributo in Atti di convegno
1996Synthesis and COMFA study of new heterocyclic compounds as potential AcylCoA: cholesterol O-acyltransferase inhibitorsContributo in Atti di convegno
1996Synthesis of 1-alkyl-3-dialkylaminoalkylamine[1]benzothieno[2,3-b]pyrazin-2(1H)-ones and their ability to antagonize KCl-induced contractions
(EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY)
Articolo in rivista
1996Transport of alpha-tocopherol and its derivatives through erythrocyte membranesContributo in Atti di convegno
1996Transport of alpha-tocopherol and its derivatives through erythrocyte membranes
(PHARMACEUTICAL RESEARCH)
Articolo in rivista
1995Isothiazoles with antiviral activityContributo in Atti di convegno
1995Nipecotic acid derivatives as potential prodrugs for brain drug deliveryContributo in Atti di convegno
1995On the reaction between 3-bromo-2-nitrobenzo[b]thiophene and some amines: a novel aromatic nucleophilic substitution with rearrangement
(JOURNAL OF THE CHEMICAL SOCIETY. PERKIN TRANSACTIONS. I)
Articolo in rivista
1995SYNTHESIS OF NOVEL 1-ALKYL OR 1-ARYL-2-(4-SUBSTITUTED-1-PIPERAZINYL)-1H-BENZOTHIENO [2,3-D]IMIDAZOLES
(JOURNAL OF HETEROCYCLIC CHEMISTRY)
Articolo in rivista
1994SYNTHESIS OF SUBSTITUTED [1]BENZOTHIENO[2,3-B]PYRAZINES AND THEIR ABILITY TO ANTAGONIZE KCL INDUCED CONTRACTIONS
(IL FARMACO)
Articolo in rivista
1993Synthesis and antifungal activity of pyrido[3',2':4,5] thieno[3,2-d]-1,2,3-triazine derivatives
(IL FARMACO)
Articolo in rivista
1992Sintesi di derivati benzotieno pirazinici potenzialmente attivi come calcio antagonistiContributo in Atti di convegno
1992Synthesis and pharmacological properties of 2-nitro-3-substituted-amino benzo[b]thiophenes and their 5-chloro derivatives
(IL FARMACO)
Articolo in rivista
1990Synthesis and pharmacological properties of 2-nitro-3-substituted-aminobenzo b thiophenes and 1-substituted benzothieno 2,3-d imidazoles
(IL FARMACO)
Articolo in rivista